Jansa, Petr

Ruzicka, Ales; Drabina, Pavel; Sedlak, Milos; Hanusek, Jiri; Valenta, Petr; Jansa, Petr, Copper(II) complexes derived from substituted 2,2′-bis-(4-isopropyl-4-methyl-4,5-dihydro-1H-imidazol-5-one) ligands: Synthesis, structure and catalytic activity. Polyhedron 2008, 27(1), 268 - 274, 10.1016/j.poly.2007.09.018 .

Sedlak, Milos; Hanusek, Jiri; Jansa, Petr; Sterba, Vojeslav, Study of ring closure reaction of substituted phenyl N-(2- thiocarbamoylphenyl)carbamates catalysed by methoxide ion. J. Phys. Org. Chem. 2006, 19(1), 61 - 67, 10.1002/poc.999 .

Hanusek, Jiri; Jansa, Petr; Russell, Mark A.; Laws, Andrew P.; Page, Michael I.; Atherton, John H.; Fettes, Kevin, Mechanism of the sulfurisation of phosphines and phosphites using 3-amino-1,2,4-dithiazole-5-thione (xanthane hydride). Organic and Biomolecular Chemistry 2007, 5(3), 478 - 484, 10.1039/b616298c .

Holy, Antonin; Jansa, Petr; Votruba, Ivan; Masojidkova, Milena; Tloust'Ova, Eva; Hrebabecky, Hubert; Horska, Kveta; Nencka, Radim, Discovery of 5-substituted-6-chlorouracils as efficient inhibitors of human thymidine phosphorylase. Journal of Medicinal Chemistry 2007, 50(24), 6016 - 6023, 10.1021/jm070644i .

Budesinsky, Milos; Holy, Antonin; Dracinsky, Martin; Jansa, Petr; Kovackova, Sona, Isotopic exchange of hydrogen at C-5 in pyrimidine derivatives: tautomers with an sp-hybridised C-5 carbon atom. European Journal of Organic Chemistry 2009(24), 4117 - 4122, 10.1002/ejoc.200900529 .

Holy, Antonin; Dracinsky, Martin; Jansa, Petr; Janeba, Zlatko; Sala, Michal; Cechova, Lucie, The optimized microwave-assisted decomposition of formamides and its synthetic utility in the amination reactions of purines. Tetrahedron 2011, 67(5), 866 - 871, 10.1016/j.tet.2010.12.040 .

Holy, Antonin; Dracinsky, Martin; Jansa, Petr; Chocholouasova, Jana; Vacek, Jaroslav; Kovackova, Soaa, Mechanism of the isotopic exchange reaction of the 5-H hydrogen of uracil derivatives in water and nonprotic solvents. European Journal of Organic Chemistry 2011(4), 777 - 785, 10.1002/ejoc.201001335 .

Holy, Antonin; Dracinsky, Martin; Jansa, Petr; Votruba, Ivan; Balzarini, Jan; Klepetarova, Blanka; Clercq, Erik de; Janeba, Zlatko; Baszczynski, Ondrej, Synthesis and antiviral activity of N-[3-fluoro-2- (phosphonomethoxy)propyl] analogues derived from N-substituted adenines and 2,6-diaminopurines. Bioorganic and Medicinal Chemistry 2011, 19(7), 2114 - 2124, 10.1016/j.bmc.2011.02.050 .

Holy, Antonin; Dracinsky, Martin; Jansa, Petr; Cesnek, Michal; Janeba, Zlatko; Baszczynski, Ondrej, Efficient and 'green' microwave-assisted synthesis of haloalkylphosphonates via the Michaelis-Arbuzov reaction. Green Chemistry 2011, 13(4), 882 - 888, 10.1039/c0gc00509f .

Holy, Antonin; Dracinsky, Martin; Jansa, Petr; Votruba, Ivan; Mackman, Richard; Cihlar, Tomas; Bahador, Gina; Janeba, Zlatko; Zidek, Zdenek; Baszczynski, Ondrej; Stepan, George, A novel and efficient one-pot synthesis of symmetrical diamide (bis-amidate) prodrugs of acyclic nucleoside phosphonates and evaluation of their biological activities. European Journal of Medicinal Chemistry 2011, 46(9), 3748 - 3754, 10.1016/j.ejmech.2011.05.040 .

Holy, Antonin; Dracinsky, Martin; Jansa, Petr; Balzarini, Jan; Klepetarova, Blanka; Janeba, Zlatko; Baszczynski, Ondrej; Hradil, Ondrej, An efficient microwave-assisted synthesis and biological properties of polysubstituted pyrimidinyl- and 1,3,5-triazinylphosphonic acids. Tetrahedron 2012, 68(3), 865 - 871, 10.1016/j.tet.2011.11.040 .

Holy, Antonin; Dracinsky, Martin; Jansa, Petr; Mertlikova-Kaiserova, Helena; Prochazkova, Eliska, Determination of the antioxidative activity of substituted 5-aminopyrimidines. Free Radical Research 2012, 46(1), 61 - 67, 10.3109/10715762.2011.638292 .

Krecmerova, Marcela; Holy, Antonin; Jansa, Petr; Otmar, Miroslav; Baszczynski, Ondrej; Blazek, Jiri; Kaiser, Martin Maxmilian; Drancinsky, Martin; Kralova, Blanka, An enzymatic glycosylation of nucleoside analogues using β-galactosidase from Escherichia coli. Bioorganic and Medicinal Chemistry 2012, 20(9), 3111 - 3118, 10.1016/j.bmc.2012.02.062 .

Holy, Antonin; Dracinsky, Martin; Jansa, Petr; Cechova, Lucie; Mertlikova-Kaiserova, Helena; Prochazkova, Eliska; Brezinova, Anna, Compound instability in dimethyl sulphoxide, case studies with 5-aminopyrimidines and the implications for compound storage and screening. Bioorganic and Medicinal Chemistry Letters 2012, 22(20), 6405 - 6409, 10.1016/j.bmcl.2012.08.065 .

Holy, Antonin; Dracinsky, Martin; Jansa, Petr; Hockova, Dana; Janeba, Zlatko; Keough, Dianne T.; Guddat, Luke W.; Baszczynski, Ondrej, The effect of novel [3-fluoro-(2-phosphonoethoxy)propyl]purines on the inhibition of Plasmodium falciparum, Plasmodium vivax and human hypoxanthine-guanine-(xanthine) phosphoribosyltransferases. European Journal of Medicinal Chemistry 2013, 67, 81 - 89, 10.1016/j.ejmech.2013.06.032 .

Dracinsky, Martin; Jansa, Petr; Janeba, Zlatko; Mertlikova-Kaiserova, Helena; Kolman, Viktor; Kostinova, Alexandra, Efficient synthesis and biological properties of the 2'-trifluoromethyl analogues of acyclic nucleosides and acyclic nucleoside phosphonates. Collect. Czech. Chem. Commun. 2011, 76(10), 1187 - 1198, 10.1135/cccc2011105 .

Dracinsky, Martin; Jansa, Petr; Votruba, Ivan; Klepetarova, Blanka; Janeba, Zlatko; Brehova, Petra; Spacek, Petr, Efficient one-pot synthesis of polysubstituted 6-[(1H-1,2,3-Triazol-1-Yl) Methyl]uracils through the "click" protocol. Collect. Czech. Chem. Commun. 2011, 76(9), 1121 - 1131, 10.1135/cccc2011074 .

Dracinsky, Martin; Jansa, Petr; Janeba, Zlatko; Kaiser, Martin Maxmilian, A novel type of acyclic nucleoside phosphonates derived from 2-(phosphonomethoxy)propanoic acid. Tetrahedron 2012, 68(21), 4003 - 4012, 10.1016/j.tet.2012.03.066 .

Dracinsky, Martin; Jansa, Petr; Janeba, Zlatko; Baszczynski, Ondrej; Prochazkova, Eliska, Microwave-assisted hydrolysis of phosphonate diesters: An efficient protocol for the preparation of phosphonic acids. Green Chemistry 2012, 14(8), 2282 - 2288, 10.1039/c2gc35547g .

Jansa, Petr; Janeba, Zlatko; Drainsky, Martin; Kaiser, Martin Maxmilian; Baszczynski, Ondej; Spaek, Petr, An efficient oxa-Michael addition to diethyl vinylphosphonate under mild reaction conditions. RSC Advances 2012, 2(4), 1282 - 1284, 10.1039/c2ra00938b .

Krecmerova, Marcela; Dracinsky, Martin; Jansa, Petr; Janeba, Zlatko; Neyts, Johan; Kasicka, Vaclav; Stepan, George; Sazelova, Petra; Auwerx, Joeri; Kiss, Eleonora; Goris, Nesya, 9-[2-(R)-(Phosphonomethoxy)propyl]-2,6-diaminopurine (R)-PMPDAP and its prodrugs: Optimized preparation, including identification of by-products formed, and antiviral evaluation in vitro. Bioorganic and Medicinal Chemistry 2013, 21(5), 1199 - 1208, 10.1016/j.bmc.2012.12.044 .

Dracinsky, Martin; Jansa, Petr; Janeba, Zlatko; Cechova, Lucie, A conversion of aromatic thiocyanates into sulfothioates: New synthetic route to aromatic Bunte salts. RSC Advances 2013, 3(8), 2650 - 2654, 10.1039/c2ra21975a .

Machacek, Vladimir; Jansa, Petr; Bertolasi, Valerio, Derivatives of 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid. Heterocycles 2006, 68(1), 59 - 69, 10.3987/COM-05-10571 .

Machacek, Vladimir; Jansa, Petr; Bertolasi, Valerio; Wsol, Vladimir, Hydantoins and thiohydantoins derived from 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid. Heterocycles 2006, 68(12), 2527 - 2547.

Machacek, Vladimir; Jansa, Petr; Svobodova, Marketa; Wsol, Vladimir; Nachtigall, Petr, Coordination compounds based on 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid. Molecules 2007, 12(5), 1064 - 1079, 10.3390/12051064 .

Ruzicka, Ales; Machacek, Vladimir; Jansa, Petr; Svobodova, Marketa; Prikryl, Josef; Cerny, Michal; Nachtigall, Petr, Stable triazenes derived from 2-alkylaminonaphthalenes and 5-nitrobenzo[c]-1,2-thiazole-3-diazonium hydrogensulfate. European Journal of Organic Chemistry 2008(19), 3272 - 3278, 10.1002/ejoc.200800180 .

Holy, Antonin; Jansa, Petr; Cesnek, Michal, METHOD OF THE SYNTHESIS OF DIALKYL HALOALKYLPHOSPHONATES AND DIALKYL HALOALKYLOXYALKYLPHOSPHONATES, WO2012/13168, 2012.

Holy, Antonin; Jansa, Petr; Janeba, Zlatko; Zidek, Zdenek; Kmonickova, Eva, PYRIMIDINE COMPOUNDS INHIBITING THE FORMATION OF NITRIC OXIDE AND PROSTAGLANDIN E2, METHOD OF PRODUCTION THEREOF AND USE THEREOF, WO2012/116666, 2012.