Masojidkova, Milena
Articles
Holy, Antonin;
Hocek, Michal;
Masojidkova, Milena, SYNTHESIS OF ACYCLIC NUCLEOTIDE ANALOGUES DERIVED FROM 2-(AMINOMETHYL)ADENINE AND 2-(AMINOMETHYL)HYPOXANTHINE. Collect. Czech. Chem. Commun. 1995, 60(5), 875 - 882, 10.1135/cccc19950875 
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Holy, Antonin;
Hocek, Michal;
Masojidkova, Milena;
Andrei, Graciela;
Snoeck, Robert;
Balzarini, Jan;
De Clercq, Erik, Synthesis and antiviral activity of acyclic nucleotide analogues derived from 6-(aminomethyl)purines and purine-6-carboxamidines. Collect. Czech. Chem. Commun. 1996, 61(10), 1525 - 1537, 10.1135/cccc19961525 .
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Holy, Antonin;
Hocek, Michal;
Masojidkova, Milena, Synthesis of acyclic nucleotide analogues derived from N-substituted 6-(1-aminoethyl)purines via 6-acetylpurine derivatives. Tetrahedron 1997, 53(6), 2291 - 2302, 10.1016/S0040-4020(96)01130-1 .
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Holy, Antonin;
Hocek, Michal;
Masojidkova, Milena, Synthesis of acyclic nucleotide analogues derived from 6-hetarylpurines via cross-coupling reactions of 9-[2-(diethoxyphosphonylmethoxy)ethyl]-6-iodopurine with hetaryl organometallic reagents. Collect. Czech. Chem. Commun. 1997, 62(1), 136 - 146.
Holy, Antonin;
Masojidkova, Milena;
Rosenberg, Ivan, PHOSPHONYLMETHOXYALKYL AND PHOSPHONYLALKYL DERIVATIVES OF ADENINE. Collect. Czech. Chem. Commun. 1988, 53(11B), 2753 - 2777.
Holy, Antonin;
Dvorakova, Hana;
Masojidkova, Milena, FLUORESCENT ANALOGUES OF ACYCLIC INHIBITORS OF S-ADENOSYL-L-HOMOCYSTEINE HYDROLASE. Collect. Czech. Chem. Commun. 1988, 53(8), 1779 - 1794.
Budesinsky, Milos;
Holy, Antonin;
Masojidkova, Milena;
Rosenberg, Ivan;
Zajicek, Jaroslav, CONFORMATIONAL STUDY ON RIBONUCLEOSIDE O-PHOSPHONYLMETHYL DERIVATIVES BY 1H NMR SPECTROSCOPY. Collect. Czech. Chem. Commun. 1985, 50(8), 1899 - 1905.
Holy, Antonin;
Masojidkova, Milena;
Spassova, Maria K., RIBONUCLEOSIDES OF 3-AMINO- AND 3,5-DIAMINOPYRAZOLE-4-CARBOXYLIC ACID AND THEIR OPEN-CHAIR ANALOGUES: SYNTHESIS AND REACTIONS. Collect. Czech. Chem. Commun. 1986, 51(7), 1512 - 1531.
Krecmerova, Marcela;
Holy, Antonin;
Masojidkova, Milena;
Hrebabecky, Hubert, PREPARATION OF PURINE 2'-DEOXY-5'-O-PHOSPHONOMETHYLNUCLEOSIDES AND 2'-DEOXY-3'-O-PHOSPHONOMETHYLNUCLEOSIDES. Collect. Czech. Chem. Commun. 1993, 58(2), 421 - 434, 10.1135/cccc19930421 .
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Holy, Antonin;
Dvorakova, Hana;
Votruba, Ivan;
Masojidkova, Milena, SYNTHESIS AND BIOLOGICAL EFFECTS OF ACYCLIC ANALOGS OF DEAZAPURINE NUCLEOSIDES. Collect. Czech. Chem. Commun. 1993, 58(3), 629 - 648, 10.1135/cccc19930629 .
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Holy, Antonin;
Masojidkova, Milena;
Otmar, Miroslav;
Rosenberg, Ivan, <5-(ADENIN-9-YL)-5-DEOXYPENTOFURANOSYL>PHOSPHONATES - A NOVEL TYPE NUCLEOTIDE ANALOGS RELATED TO HPMPA. I. DERIVATIVES WITH L-arabino, D-arabino, 2-DEOXY-L-erythro AND 2-DEOXY-L-threo CONFIGURATION. Collect. Czech. Chem. Commun. 1993, 58(9), 2159 - 2179, 10.1135/cccc19932159 .
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Holy, Antonin;
Masojidkova, Milena;
Otmar, Miroslav;
Rosenberg, Ivan, <5-(ADENIN-9-YL)-5-DEOXY-L-PENTOFURANOSYL>PHOSPHONATES - A NOVEL TYPE OF NUCLEOTIDE ANALOGS RELATED TO HPMPA. II. SYNTHESIS OF L-ribo and L-xylo CONFIGURATED DERIVATIVES BY RECYCLIZATION OF DIETHYL (5-RS)-<1,2-O-ISOPROPYLIDENE-5-O-METHANESULFONYL-D-PENTOFURANOS-5-C-YL>PHOSPHONATES .... Collect. Czech. Chem. Commun. 1993, 58(9), 2180 - 2196, 10.1135/cccc19932180 .
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Budesinsky, Milos;
Holy, Antonin;
Dvorakova, Hana;
Masojidkova, Milena;
Spassova, Maria, SYNTHEIS OF N-(3-AZIDO-2-HYDROXYPROPYL), N-(3-PHTHALIMIDO-2-HYDROXYPROPYL) AND N-(3-AMINO-2-HYDROXYPROPYL)DERIVATIVES OF HETEROCYCLIC BASES. Collect. Czech. Chem. Commun. 1994, 59(5), 1153 - 1174, 10.1135/cccc19941153 .
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Holy, Antonin;
Masojidkova, Milena;
Alexander, Petr, PREPARATION OF 9-(2-PHOSPHONOMETHOXYETHYL)ADENINE ESTERS AS POTENTIAL PRODRUGS. Collect. Czech. Chem. Commun. 1994, 59(8), 1853 - 1869, 10.1135/cccc19941853 .
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Holy, Antonin;
Masojidkova, Milena;
Alexander, Petr, SYNTHESIS OF 9-(2-PHOSPHONOMETHOXYETHYL)ADENINE AND RELATED COMPOUNDS. Collect. Czech. Chem. Commun. 1994, 59(8), 1870 - 1878, 10.1135/cccc19941870 .
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Budesinsky, Milos;
Holy, Antonin;
Masojidkova, Milena;
Hockova, Dana, ACYCLIC NUCLEOSIDE AND NUCLEOTIDE ANALOGS DERIVED FROM 2-AZAADENINE. Collect. Czech. Chem. Commun. 1995, 60(2), 224 - 236, 10.1135/cccc19950224 .
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Krecmerova, Marcela;
Holy, Antonin;
Masojidkova, Milena, SYNTHESIS OF 3-(4-PYRIDINYL)-, 3-(2-CHLORO-4-PYRIDINYL)- AND 3-(2-AMINO-4-PYRIDINYL)PROPOXYMETHANEPHOSPHONIC ACID. Collect. Czech. Chem. Commun. 1995, 60(4), 670 - 680, 10.1135/cccc19950670 .
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Holy, Antonin;
Masojidkova, Milena, SYNTHESIS OF ENANTIOMERIC N-(2-PHOSPHONOMETHOXYPROPYL) DERIVATIVES OF PURINE AND PYRIMIDINE BASES. I. THE STEPWISE APPROACH. Collect. Czech. Chem. Commun. 1995, 60(7), 1196 - 1212, 10.1135/cccc19951196 .
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Holy, Antonin;
Dvorakova, Hana;
Masojidkova, Milena, SYNTHESIS OF ENANTIOMERIC N-(2-PHOSPHONOMETHOXYPROPYL)DERIVATIVES OF PURINE AND PYRIMIDINE BASES. II. THE SYNTHON APPROACH. Collect. Czech. Chem. Commun. 1995, 60(8), 1390 - 1409, 10.1135/cccc19951390 .
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Holy, Antonin;
Masojidkova, Milena;
Votavova, Hana;
Janeba, Zlatko, Intramolecular cyclization of some acyclic nucleoside analogs. Collect. Czech. Chem. Commun. 1996, 61(3), 442 - 457, 10.1135/cccc19960442 .
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Krecmerova, Marcela;
Holy, Antonin;
Masojidkova, Milena;
Hrebabecky, Hubert, Synthesis of 5-phenyl-2(1H)-pyrimidinone nucleosides. Collect. Czech. Chem. Commun. 1996, 61(3), 458 - 477, 10.1135/cccc19960458 .
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Krecmerova, Marcela;
Holy, Antonin;
Masojidkova, Milena;
Hrebabecky, Hubert, 2′,3′-dideoxy- and 3′-azido-2′,3′-dideoxynucleosides of 5-phenyl-2(1H)-pyrimidinone. Preparation of 2′,3′-dideoxypentofuranoses. Collect. Czech. Chem. Commun. 1996, 61(3), 478 - 488, 10.1135/cccc19960478 .
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Holy, Antonin;
Dvorakova, Hana;
Masojidkova, Milena;
Andrei, Graciela;
Snoeck, Robert;
Balzarini, Jan;
De Clercq, Erik, Synthesis of 2'-aminomethyl derivatives of N-(2- (phosphonomethoxy)ethyl) nucleotide analogues as potential antiviral agents. Journal of Medicinal Chemistry 1996, 39(17), 3263 - 3268, 10.1021/jm9601314 .
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Budesinsky, Milos;
Holy, Antonin;
Jindrich, Jindrich;
Dvorakova, Hana;
Masojidkova, Milena;
Balzarini, Jan;
De Clercq, Erik;
Andrei, Graciella, Acyclic nucleotide analogs derived from 8-azapurines: Synthesis and antiviral activity. Journal of Medicinal Chemistry 1996, 39(20), 4073 - 4088, 10.1021/jm960314q .
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Holy, Antonin;
Masojidkova, Milena;
Hockova, Dana, "Abbreviated" NADanalogues containing a phosphonate function. Collect. Czech. Chem. Commun. 1996, 61(10), 1538 - 1548, 10.1135/cccc19961538 .
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Holy, Antonin;
Masojidkova, Milena;
Otmar, Miroslav, Two Synthetic Approaches to 9-Deaza Analogues of 9-(2,3-Dihydroxypropyl)adenine (DHPA). Collect. Czech. Chem. Commun. 1996, 61, S49 - S51.
Budesinsky, Milos;
Holy, Antonin;
Masojidkova, Milena;
Hrebabecky, Hubert;
Havlas, Zdenek, 1-(3,5-O-alkylidene-2-deoxy-4-C-hydroxymethyl-α-L-threo- pentofuranosyl)uracils. Collect. Czech. Chem. Commun. 1997, 62(6), 957 - 970.
Holy, Antonin;
Masojidkova, Milena;
Hrebabecky, Hubert, Synthesis of carba analogues of deoxy-4-C-(hydroxymethyl)-pentofuranoses, intermediates in the synthesis of carbocyclic nucleosides. Collect. Czech. Chem. Commun. 1998, 63(12), 2044 - 2064.
Holy, Antonin;
Dvorakova, Hana;
Masojidkova, Milena;
Andrei, Graciela;
Snoeck, Robert;
Balzarini, Jan;
De Clercq, Erik;
Guenter, Jaroslav, Structure-antiviral activity relationship in the series of pyrimidine and purine N-[2-(2-phosphonomethoxy)ethyl] nucleotide analogues. 1. Derivatives substituted at the carbon atoms of the base. Journal of Medicinal Chemistry 1999, 42(12), 2064 - 2086, 10.1021/jm9811256 .
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Holy, Antonin;
Masojidkova, Milena;
Meszarosova, Katerina, Synthesis of acyclic adenine 8,N-anhydronucleosides. Collect. Czech. Chem. Commun. 2000, 65(7), 1109 - 1125.
Holy, Antonin;
Masojidkova, Milena;
Janeba, Zlatko, Synthesis of acyclic nucleoside and nucleotide analogs derived from 6-amino-7H-purin-8(9H)-one. Collect. Czech. Chem. Commun. 2000, 65(7), 1126 - 1144.
Holy, Antonin;
Masojidkova, Milena;
Janeba, Zlatko, Synthesis of acyclic nucleoside and nucleotide analogs derived from 6-amino-7H-purine-8(9H)-thione and 8-(methylsulfanyl)adenine. Collect. Czech. Chem. Commun. 2000, 65(11), 1698 - 1712.
Budesinsky, Milos;
Holy, Antonin;
Masojidkova, Milena;
Alexander, Petr, Synthesis of acyclic nucleotide analogues derived from N-substituted isoguanine. Collect. Czech. Chem. Commun. 2000, 65(11), 1713 - 1725.
Holy, Antonin;
Votruba, Ivan;
Masojidkova, Milena;
Otmar, Miroslav, An alternative synthesis of HPMPC and HPMPA diphosphoryl derivatives. Collect. Czech. Chem. Commun. 2001, 66(3), 500 - 506, 10.1135/cccc20010500 .
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Holy, Antonin;
Masojidkova, Milena;
Otmar, Miroslav;
Polakova, Lucie, A facile synthesis of azetidin-2-ylphosphonic acid and its 1-alkyl derivatives. Collect. Czech. Chem. Commun. 2001, 66(3), 507 - 516, 10.1135/cccc20010507 .
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Holy, Antonin;
Masojidkova, Milena;
Janeba, Zlatko, Synthesis of 8-amino-and N-substituted 8-aminoadenine derivatives of acyclic nucleoside and nucleotide analogs. Collect. Czech. Chem. Commun. 2001, 66(3), 517 - 532, 10.1135/cccc20010517 .
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Holy, Antonin;
Masojidkova, Milena;
Janeba, Zlatko, Transformation of 8-[(2-hydroxyalkyl)sulfanyl]adenines to 6-amino-7H-purin-8(9H)-one derivatives. Collect. Czech. Chem. Commun. 2001, 66(9), 1393 - 1406, 10.1135/cccc20011393 .
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Holy, Antonin;
Votruba, Ivan;
Masojidkova, Milena;
Tloustova, Eva, Synthesis and cytostatic activity of N-[2-(phosphonomethoxy)alkyl] derivatives of N-substituted adenines, 2,6-diaminopurines and related compounds. Collect. Czech. Chem. Commun. 2001, 66(10), 1545 - 1592.
Holy, Antonin;
Cesnek, Michal;
Masojidkova, Milena, 6-Guanidinopurine nucleosides and their analogues. Tetrahedron 2002, 58(15), 2985 - 2996, 10.1016/S0040-4020(02)00186-2 .
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Holy, Antonin;
Votruba, Ivan;
Masojidkova, Milena;
Andrei, Graciela;
Snoeck, Robert;
Balzarini, Jan;
De Clercq, Erik;
Naesens, Lieve, 6-[2-(Phosphonomethoxy)alkoxy]pyrimidines with antiviral activity. Journal of Medicinal Chemistry 2002, 45(9), 1918 - 1929, 10.1021/jm011095y .
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Holy, Antonin;
Masojidkova, Milena;
Hrebabecky, Hubert, Synthesis of racemic 2-hydroxy-4- and 2-hydroxy-5-(hydroxymethyl)cyclohexane nucleoside analogues. Collect. Czech. Chem. Commun. 2002, 67(11), 1681 - 1699, 10.1135/cccc20021681 .
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Holy, Antonin;
Votruba, Ivan;
Masojidkova, Milena;
Capek, Petr;
Otmar, Miroslav, A facile synthesis of 9-deaza analogue of olomoucine. Collect. Czech. Chem. Commun. 2003, 68(4), 779 - 791, 10.1135/cccc20030779 .
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Budesinsky, Milos;
Krecmerova, Marcela;
Holy, Antonin;
Masojidkova, Milena, Synthesis of optically active N-alkyl derivatives of (R)-3-(adenin-9-yl)-2-hydroxypropanoic acid and related compounds. Collect. Czech. Chem. Commun. 2003, 68(5), 931 - 950, 10.1135/cccc20030931 .
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Holy, Antonin;
Masojidkova, Milena;
Andrei, Graciela;
Snoeck, Robert;
Balzarini, Jan;
De Clercq, Erik;
Hockova, Dana, 5-Substituted-2,4-diamino-6-[2-(phosphonomethoxy) ethoxy]pyrimidines-Acyclic Nucleoside Phosphonate Analogues with Antiviral Activity. Journal of Medicinal Chemistry 2003, 46(23), 5064 - 5073.
Holy, Antonin;
Cesnek, Michal;
Masojidkova, Milena, New 2-alkynyl derivatives of the acyclic nucleoside 9-(2,3-dihydroxypropyl) adenine and their 6-guanidinopurine counterparts as potential effectors of adenosine receptors. Collect. Czech. Chem. Commun. 2003, 68(11), 2201 - 2218, 10.1135/cccc20032201 .
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Holy, Antonin;
Masojidkova, Milena;
Hrebabecky, Hubert;
Sala, Michal, Synthesis of racemic 2-hydroxy-4- and 2-hydroxy-5-(hydroxymethyl) cyclohexane pyrimidine C-Nucleoside analogues. Collect. Czech. Chem. Commun. 2004, 69(4), 918 - 932, 10.1135/cccc20040918 .
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Holy, Antonin;
Votruba, Ivan;
Masojidkova, Milena;
Hockova, Dana, An efficient synthesis of cytostatic mono and bis-alkynylpyrimidine derivatives by the Sonogashira cross-coupling reactions of 2,4-diamino-6- iodopyrimidine and 2-amino-4,6-dichloropyrimidine. Tetrahedron 2004, 60(23), 4983 - 4987, 10.1016/j.tet.2004.04.035 .
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Holy, Antonin;
Masojidkova, Milena;
Hrebabecky, Hubert, Synthesis of purine nucleoside analogues derived from carbocyclic 5-C-(hydroxymethyl)hexopyranoses. Collect. Czech. Chem. Commun. 2004, 69(2), 435 - 452.
Krecmerova, Marcela;
Holy, Antonin;
Masojidkova, Milena, Synthesis of N- and N-[2-hydroxy-3- (phosphonomethoxy)-propyl] derivatives of N-substituted adenines, 2,6-diaminopurines and related compounds. Collect. Czech. Chem. Commun. 2004, 69(10), 1889 - 1913, 10.1135/cccc20041889 .
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Holy, Antonin;
Masojidkova, Milena;
Zidek, Zdenek;
Kmonickova, Eva;
Dolakova, Petra, Synthesis and immunobiological activity of base substituted 2-amino-3-(purin-9-yl)propanoic acid derivatives. Bioorganic and Medicinal Chemistry 2005, 13(7), 2349 - 2354, 10.1016/j.bmc.2005.01.054 .
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Holy, Antonin;
Masojidkova, Milena;
Hockova, Dana, Sonogashira cross-coupling in the synthesis of acyclic nucleoside phosphonates: Preparation of 6-[(phosphonomethoxy)alkynyl]- and 6-[(phosphonomethoxy)alkyl]pyrimidines. Collect. Czech. Chem. Commun. 2005, 70(2), 247 - 258, 10.1135/cccc20050247 .
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Holy, Antonin;
Masojidkova, Milena;
Hrebabecky, Hubert, Synthesis of racemic 9-(6- and 2,6-substituted 9H-purin-9-yl)-5- oxatricyclo[4.2.1.0]nonane-3-methanols, novel conformationally locked carbocyclic nucleosides. Collect. Czech. Chem. Commun. 2005, 70(1), 103 - 123, 10.1135/cccc20050103 .
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Holy, Antonin;
Cesnek, Michal;
Masojidkova, Milena;
Zidek, Zdenek, Synthesis of 9-alkyl and 9-heteroalkyl substituted 2-amino-6- guanidinopurines and their influence on the NO-production in macrophages. Bioorganic and Medicinal Chemistry 2005, 13(8), 2917 - 2926, 10.1016/j.bmc.2005.02.008 .
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Holy, Antonin;
Masojidkova, Milena;
Dolakova, Petra, Synthesis of Base Substituted 2-Hydroxy-3-(purin-9-yl)-propanoic Acids and 4-(Purin-9-yl)-3-butenoic Acids. Nucleosides, Nucleotides and Nucleic Acids 2003, 22(12), 2145 - 2160, 10.1081/NCN-120026636 .
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Holy, Antonin;
Votruba, Ivan;
Masojidkova, Milena;
Tloust'Ova, Eva;
Hrebabecky, Hubert;
Horska, Kveta;
Nencka, Radim, Design and synthesis of novel 5,6-disubstituted uracil derivatives as potent inhibitors of thymidine phosphorylase. Bioorganic and Medicinal Chemistry Letters 2006, 16(5), 1335 - 1337, 10.1016/j.bmcl.2005.11.050 .
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Holy, Antonin;
Masojidkova, Milena;
Hrebabecky, Hubert, Synthesis of novel conformationally locked carbocyclic nucleosides derived from 5,5- and 6,6-bis(hydroxymethyl)bicyclo[2.2.1]heptan-2-ol. Collect. Czech. Chem. Commun. 2005, 70(4), 519 - 538, 10.1135/cccc20050519 .
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Holy, Antonin;
Votruba, Ivan;
Masojidkova, Milena;
Otmar, Miroslav, Synthesis and antiproliferative activity of 2,6-diamino-9-benzyl-9- deazapurine and related compounds. Bioorganic and Medicinal Chemistry 2004, 12(12), 3187 - 3195, 10.1016/j.bmc.2004.04.003 .
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Holy, Antonin;
Masojidkova, Milena;
Andrei, Graciela;
Snoeck, Robert;
Balzarini, Jan;
De Clercq, Erik;
Hockova, Dana, Synthesis and antiviral activity of 2,4-diamino-5-cyano-6-[2- (phosphonomethoxy)ethoxy]pyrimidine and related compounds. Bioorganic and Medicinal Chemistry 2004, 12(12), 3197 - 3202, 10.1016/j.bmc.2004.04.002 .
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Holy, Antonin;
Masojidkova, Milena;
Pohl, Radek;
Otmar, Miroslav;
Bambuch, Vitezslav, C-Functionalization of 9-deazapurines by cross-coupling reactions. Tetrahedron 2007, 63(7), 1589 - 1601, 10.1016/j.tet.2006.12.008 .
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Holy, Antonin;
Masojidkova, Milena;
Chalupova, Sarka, Synthesis of some N-substituted derivatives of 1-[(S)-3-hydroxy-2-(phosphonomethoxy)propyl]cytosine (HPMPC, cidofovir). Collect. Czech. Chem. Commun. 2005, 70(12), 2053 - 2065, 10.1135/cccc20052053 .
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Holy, Antonin;
Masojidkova, Milena;
Chalupova, Sarka, Synthesis of N-substituted derivatives of 1-[2- (phosphonomethoxy)ethyl]cytosine and its diisopropyl ester as a model reaction for the synthesis of N-substituted derivatives of cidofovir. Collect. Czech. Chem. Commun. 2005, 70(12), 2066 - 2074, 10.1135/cccc20052066 .
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Holy, Antonin;
Masojidkova, Milena;
Pohl, Radek;
Vrbovska, Silvie, Bifunctional acyclic nucleoside phosphonates. 1. Symmetrical 1,3-bis[(phosphonomethoxy)propan-2-yl] derivatives of purines and pyrimidines. Collect. Czech. Chem. Commun. 2006, 71(4), 543 - 566, 10.1135/cccc20060543 .
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Krecmerova, Marcela;
Holy, Antonin;
Masojidkova, Milena, Preparation of C-5 substituted cidofovir derivatives. Collect. Czech. Chem. Commun. 2006, 71(4), 579 - 594, 10.1135/cccc20060579 .
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Krecmerova, Marcela;
Holy, Antonin;
Masojidkova, Milena;
Andrei, Graciela;
Snoeck, Robert;
Balzarini, Jan;
De Clercq, Erik;
Naesens, Lieve;
Piskala, Alois;
Neyts, Johan, Antiviral activity of triazine analogues of 1-(S)-[3-hydroxy-2- (phosphonomethoxy)propyl]cytosine (cidofovir) and related compounds. Journal of Medicinal Chemistry 2007, 50(5), 1069 - 1077, 10.1021/jm061281+ .
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Holy, Antonin;
Masojidkova, Milena;
Hrebabecky, Hubert;
Sala, Michal, Synthesis of novel racemic conformationally locked carbocyclic nucleosides derived from 7-substituted bicyclo[2.2.1]hept-5-ene-2,2-dimethanols. Collect. Czech. Chem. Commun. 2006, 71(5), 635 - 649, 10.1135/cccc20060635 .
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Holy, Antonin;
Dracinsky, Martin;
Masojidkova, Milena;
Hrebabecky, Hubert, Synthesis of novel conformationally locked carbocyclic nucleosides derived from 3-(hydroxymethyl)bicyclo[2.2.1]heptane-2,5-diol. Collect. Czech. Chem. Commun. 2006, 71(6), 871 - 888, 10.1135/cccc20060871 .
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Holy, Antonin;
Masojidkova, Milena;
Dolakova, Petra, Efficient synthesis of pyrimidinecarbonitriles and their derivatives. Heterocycles 2007, 71(5), 1107 - 1115.
Krecmerova, Marcela;
Holy, Antonin;
Masojidkova, Milena;
Andrei, Graciela;
Snoeck, Robert;
Balzarini, Jan;
De Clercq, Erik;
Pohl, Radek;
Naesens, Lieve;
Neyts, Johan, Ester prodrugs of cyclic 1-(S)-[3-hydroxy-2-(phosphonomethoxy)propyl]-5- azacytosine: Synthesis and antiviral activity. Journal of Medicinal Chemistry 2007, 50(23), 5765 - 5772, 10.1021/jm0707166 .
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Holy, Antonin;
Cesnek, Michal;
Masojidkova, Milena;
Solinova, Veronika;
Koval, Dusan;
Kasicka, Vaclav, Synthesis and properties of 2-guanidinopurines. Collect. Czech. Chem. Commun. 2006, 71(9), 1303 - 1319, 10.1135/cccc20061303 .
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Holy, Antonin;
Cesnek, Michal;
Masojidkova, Milena;
Zidek, Zdenek;
Kmonickova, Eva, Synthesis of guanidino analogues of PMPDAP and their immunobiological activity. Bioorganic and Medicinal Chemistry 2008, 16(2), 965 - 980, 10.1016/j.bmc.2007.10.010 .
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Holy, Antonin;
Jansa, Petr;
Votruba, Ivan;
Masojidkova, Milena;
Tloust'Ova, Eva;
Hrebabecky, Hubert;
Horska, Kveta;
Nencka, Radim, Discovery of 5-substituted-6-chlorouracils as efficient inhibitors of human thymidine phosphorylase. Journal of Medicinal Chemistry 2007, 50(24), 6016 - 6023, 10.1021/jm070644i .
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Krecmerova, Marcela;
Holy, Antonin;
Masojidkova, Milena, Pyrimidine acyclic nucleotide analogues with aromatic substituents in C-5 position. Collect. Czech. Chem. Commun. 2007, 72(7), 927 - 951, 10.1135/cccc20070927 .
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Holy, Antonin;
Dracinsky, Martin;
Masojidkova, Milena;
Dolakova, Petra;
Solinova, Veronika;
Kasicka, Vaclav, Acyclic nucleoside bisphosphonates: Synthesis and properties of chiral 2-amino-4,6-bis[(phosphonomethoxy)alkoxy]pyrimidines. European Journal of Medicinal Chemistry 2009, 44(6), 2408 - 2424, 10.1016/j.ejmech.2008.09.031 .
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Holy, Antonin;
Dracinsky, Martin;
Masojidkova, Milena;
Hrebabecky, Hubert;
Sala, Michal;
Neyts, Johan;
De Palma, Armando M., Norbornane as the novel pseudoglycone moiety in nucleosides. Tetrahedron 2009, 65(45), 9291 - 9299, 10.1016/j.tet.2009.09.018 .
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Krecmerova, Marcela;
Holy, Antonin;
Masojidkova, Milena, Acyclic nucleoside phosphonates with 5-azacytosine base moiety substituted in C-6 position. Bioorganic and Medicinal Chemistry 2010, 18(1), 387 - 395, 10.1016/j.bmc.2009.10.044 .
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Holy, Antonin;
Masojidkova, Milena;
Janeba, Zlatko, Alternative synthesis of 9-{3-[(diisopropoxyphosphoryl)-methoxy]-2- hydroxypropyl}adenine and its free phosphonates substituted at the c-8 position of purine base. Collect. Czech. Chem. Commun. 2010, 75(3), 371 - 381, 10.1135/cccc2009569 .
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Holy, Antonin;
Masojidkova, Milena;
Sala, Michal;
Neyts, Johan;
De Palma, Armando M.;
Hebabecky, Hubert;
Draeinsky, Martin, Synthesis of novel racemic carbocyclic nucleosides derived from 5,6-disubstituted norbornene. Collect. Czech. Chem. Commun. 2010, 75(1), 1 - 20, 10.1135/cccc2009116 .
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Krecmerova, Marcela;
Holy, Antonin;
Dracinsky, Martin;
Masojidkova, Milena;
Andrei, Graciela;
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