Pohl, Radek
Articles
Hocek, Michal;
Capek, Petr;
Pohl, Radek, A facile and efficient synthesis of (purin-6-yl)alanines. Journal of Organic Chemistry 2004, 69(23), 7985 - 7988, 10.1021/jo048812r 
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Hocek, Michal;
Pohl, Radek, Regioselectivity in cross-coupling reactions of 2,6,8-trichloro-9- (tetrahydropyran-2-yl)purine: Synthesis of 2,6,8-trisubstituted purine bases. Synthesis 2004(17), 2869 - 2876, 10.1055/s-2004-834881 .
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Cisarova, Ivana;
Hocek, Michal;
Pohl, Radek, Highly methylated purines and purinium salts as analogues of heteromines. European Journal of Organic Chemistry 2005(14), 3026 - 3030, 10.1002/ejoc.200500154 .
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Hocek, Michal;
Capek, Petr;
Pohl, Radek, Synthesis of enantiomerically pure (purin-6-yl)phenylalanines and their nucleosides, a novel type of purine-amino acid conjugates. Journal of Organic Chemistry 2005, 70(20), 8001 - 8008, 10.1021/jo051110x .
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Hocek, Michal;
Pohl, Radek;
Klepetarova, Blanka, A new modular and practical methodology for the synthesis of 4- or 3-substituted phenyl C-nucleosides. European Journal of Organic Chemistry 2005(21), 4525 - 4528, 10.1002/ejoc.200500607 .
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Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Silhar, Peter, Facile and efficient synthesis of 6-(hydroxymethyl)purines. Organic Letters 2004, 6(19), 3225 - 3228, 10.1021/ol049059r .
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Naus, Petr;
Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Furman, Phillip A.;
Tharnish, Phillip M.;
Otto, Michael J., Cytostatic 6-arylpurine nucleosides. 6. SAR in anti-HCV and cytostatic activity of extended series of 6-hetarylpurine ribonucleosides. Journal of Medicinal Chemistry 2005, 48(18), 5869 - 5873, 10.1021/jm050335x .
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Novak, Petr;
Kotora, Martin;
Hocek, Michal;
Pohl, Radek, Synthesis of C-aryldeoxyribosides by [2 + 2 + 2]-cyclotrimerization catalyzed by Rh, Ni, Co, and Ru complexes. Organic Letters 2006, 8(10), 2051 - 2054, 10.1021/ol060454m .
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Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Silhar, Peter, The first synthesis and cytostatic activity of novel 6-(fluoromethyl)purine bases and nucleosides. Organic and Biomolecular Chemistry 2005, 3(16), 3001 - 3007, 10.1039/b508122j .
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Hocek, Michal;
Pohl, Radek;
Klepetarova, Blanka;
Urban, Milan, New modular and efficient approach to 6-substituted pyridin-2-yl C-nucleosides. Journal of Organic Chemistry 2006, 71(19), 7322 - 7328, 10.1021/jo061080d .
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Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Silhar, Peter, Synthesis of 2-substituted 6-(hydroxymethyl)purine bases and nucleosides. Collect. Czech. Chem. Commun. 2005, 70(10), 1669 - 1695, 10.1135/cccc20051669 .
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Novak, Petr;
Kotora, Martin;
Hocek, Michal;
Turek, Pavel;
Pohl, Radek, Preparation of highly substituted 6-arylpurine ribonucleosides by Ni-catalyzed cyclotrimerization. Scope of the reaction. Journal of Organic Chemistry 2006, 71(23), 8978 - 8981, 10.1021/jo061485y .
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Hocek, Michal;
Pohl, Radek;
Klepetarova, Blanka;
Cerna, Igor, Direct C-H arylation of purines: Development of methodology and its use in regioselective synthesis of 2,6,8-trisubstituted purines. Organic Letters 2006, 8(23), 5389 - 5392, 10.1021/ol062324j .
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Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Kuchar, Martin, Synthesis of purines bearing functionalized C-substituents by the conjugate addition of nucleophiles to 6-vinylpurines and 6-ethynylpurines. European Journal of Organic Chemistry 2006(22), 5083 - 5098, 10.1002/ejoc.200600545 .
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Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Silhar, Peter, Synthesis and cytostatic activity of novel 6-(Difluoromethyl)purine bases and nucleosides. Synthesis 2006(11), 1848 - 1852, 10.1055/s-2006-942365 .
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Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Klepetarova, Blanka;
Silhar, Peter, Synthesis of 6-amino-, 6-methyl- and 6-aryl-2-(hydroxymethyl)purine bases and nucleosides. Collect. Czech. Chem. Commun. 2006, 71(6), 788 - 803, 10.1135/cccc20060788 .
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Hocek, Michal;
Votruba, Ivan;
Hobza, Pavel;
Pohl, Radek;
Klepetarova, Blanka;
Mabery, Eric;
Mackman, Richard;
Vrabel, Milan;
Havran, Ludek;
Fojta, Miroslav;
Rulisek, Lubomir;
Zendlova, Lucie;
Shih, I.-Hung, Purines bearing phenanthroline or bipyridine ligands and their RuII complexes in position 8 as model compounds for electrochemical DNA labeling - Synthesis, crystal structure, electrochemistry, quantum chemical calculations, cytostatic and antiviral activity. European Journal of Inorganic Chemistry 2007(12), 1752 - 1769, 10.1002/ejic.200700030 .
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Hocek, Michal;
Capek, Petr;
Pohl, Radek, Cross-coupling reactions of unprotected halopurine bases, nucleosides, nucleotides and nucleoside triphosphates with 4-boronophenylalanine in water. Synthesis of (purin-8-yl)- and (purin-6-yl)phenylalanines. Organic and Biomolecular Chemistry 2006, 4(11), 2278 - 2284, 10.1039/b604010a .
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Hocek, Michal;
Capek, Petr;
Pohl, Radek;
Vrabel, Milan;
Hasnik, Zbynek, Aqueous-phase Suzuki-Miyaura cross-coupling reactions of free halopurine bases. Synthesis 2006(20), 3515 - 3526, 10.1055/s-2006-950240 .
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Hocek, Michal;
Pohl, Radek;
Klepetarova, Blanka;
Joubert, Nicolas, Modular and practical synthesis of 6-substituted pyridin-3-yl C-nucleosides. Journal of Organic Chemistry 2007, 72(18), 6797 - 6805, 10.1021/jo0709504 .
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Hocek, Michal;
Capek, Petr;
Pohl, Radek;
Cahova, Hana;
Gloeckner, Christian;
Marx, Andreas, An efficient method for the construction of functionalized dna bearing amino acid groups through cross-coupling reactions of nucleoside triphosphates followed by primer extension or PCR. Chemistry - A European Journal 2007, 13(21), 6196 - 6203, 10.1002/chem.200700220 .
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Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Klepetarova, Blanka;
Vrabel, Milan, Synthesis of 2′-deoxyadenosine nucleosides bearing bipyridine-type ligands and their Ru-complexes in position 8 through cross-coupling reactions. Organic and Biomolecular Chemistry 2007, 5(17), 2849 - 2857, 10.1039/b709245h .
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Hocek, Michal;
Pohl, Radek;
Cerna, Igor, The first direct C-H arylation of purine nucleosides. Chemical Communications 2007(45), 4729 - 4730, 10.1039/b714253f .
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Hocek, Michal;
Pohl, Radek;
Silhar, Peter, Cytostatic and antiviral 6-arylpurine ribonucleosides VIII. Synthesis and evaluation of 6-substituted purine 3′-deoxyribonucleosides. Collect. Czech. Chem. Commun. 2006, 71(10), 1484 - 1496, 10.1135/cccc20061484 .
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Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Shih, I-hung;
Mabery, Eric;
Mackman, Richard;
Kuchar, Martin, Synthesis, cytostatic, and antiviral activity of novel 6-[2-(dialkylamino)ethyl]-, 6-(2-alkoxyethyl)-, 6-[2-(alkylsulfanyl)ethyl]-, and 6-[2-(dialkylamino)vinyl]purine nucleosides. Bioorganic and Medicinal Chemistry 2008, 16(3), 1400 - 1424, 10.1016/j.bmc.2007.10.063 .
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Hocek, Michal;
Pohl, Radek;
Klepetarova, Blanka;
Barta, Jan;
Ernsting, Nikolaus P., Modular synthesis of 5-substituted thiophen-2-yl C-2′- deoxyribonucleosides. Journal of Organic Chemistry 2008, 73(10), 3798 - 3806, 10.1021/jo800177y .
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Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Silhar, Peter;
Shih, I-hung;
Mabery, Eric;
Mackman, Richard, Synthesis, cytostatic and anti-HCV activity of 6-(N-substituted aminomethyl)-, 6-(O-substituted hydroxymethyl)- and 6-(S-substituted sulfanylmethyl)purine nucleosides. Bioorganic and Medicinal Chemistry 2008, 16(5), 2329 - 2366, 10.1016/j.bmc.2007.11.067 .
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Hocek, Michal;
Pohl, Radek;
Vrabel, Milan;
Havran, Ludek;
Fojta, Miroslav;
Brazdilova, Petra;
Pivonkova, Hana, Ferrocenylethynyl derivatives of nucleoside triphosphates: Synthesis, incorporation, electrochemistry, and bioanalytical applications. Chemistry - A European Journal 2007, 13(34), 9527 - 9533, 10.1002/chem.200701249 .
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Hocek, Michal;
Pohl, Radek;
Klepetarova, Blanka;
Kuchar, Martin, Synthesis of diverse 6-(1,2-disubstituted ethyl)purine bases and nucleosides via 6-(oxiran-2-yl)purines. Tetrahedron 2008, 64(45), 10355 - 10364, 10.1016/j.tet.2008.08.074 .
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Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Klepetarova, Blanka;
Kuchar, Martin, Synthesis of substituted 6-cyclopropylpurine bases and nucleosides by cross-coupling reactions or cyclopropanations. Organic and Biomolecular Chemistry 2008, 6(13), 2377 - 2387, 10.1039/b802833h .
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Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Vrabel, Milan;
Ernsting, Nikolaus P.;
Sajadi, Mohsen;
Kovalenko, Sergey A., Synthesis and photophysical properties of 7-deaza-2′-deoxyadenosines bearing bipyridine ligands and their Ru(ii)-complexes in position 7. Organic and Biomolecular Chemistry 2008, 6(16), 2852 - 2860, 10.1039/b805632c .
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Hocek, Michal;
Pohl, Radek;
Cahova, Hana;
Bednarova, Lucie;
Novakova, Katerina;
Cvacka, Josef, Synthesis of 8-bromo-, 8-methyl- and 8-phenyl-dATP and their polymerase incorporation into DNA. Organic and Biomolecular Chemistry 2008, 6(20), 3657 - 3660, 10.1039/b811935j .
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Hocek, Michal;
Pohl, Radek;
Havran, Ludek;
Fojta, Miroslav;
Cahova, Hana;
Brazdilova, Petra;
Pivonkova, Hana, Aminophenyl- and nitrophenyl-labeled nucleoside triphosphates: Synthesis, enzymatic incorporation, and electrochemical detection. Angewandte Chemie - International Edition 2008, 47(11), 2059 - 2062, 10.1002/anie.200705088 .
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Hocek, Michal;
Pohl, Radek;
Urban, Milan;
Joubert, Nicolas, Modular Synthesis of 4-aryl- and 4-amino-substituted benzene C-2′-Deoxyribonucleosides. Synthesis 2008(12), 1918 - 1932, 10.1055/s-2008-1067038 .
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Kotora, Martin;
Hocek, Michal;
Turek, Pavel;
Pohl, Radek;
Klepetarova, Blanka, Cobalt-induced synthesis of 6-(pyridin-2-yl)purines by microwave-enhanced [2+2+2] cyclotrimerization. European Journal of Organic Chemistry 2008(19), 3335 - 3343, 10.1002/ejoc.200800205 .
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Hocek, Michal;
Pohl, Radek;
Bambuch, Vitezslav, Synthesis of 6-(4,5-dihydrofuran-2-yl)- and 6-(tetrahydrofuran-2-yl)purine bases and nucleosides. European Journal of Organic Chemistry 2008(16), 2783 - 2788, 10.1002/ejoc.200800174 .
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Hocek, Michal;
Pohl, Radek;
Klepetarova, Blanka;
Stefko, Martin, A modular methodology for the synthesis of 4- and 3-substituted benzene and aniline C-ribonucleosides. European Journal of Organic Chemistry 2008(10), 1689 - 1704, 10.1002/ejoc.200701168 .
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Hocek, Michal;
Pohl, Radek;
Klepetarova, Blanka;
Cerna, Igor, Synthesis of 6,8,9-tri- and 2,6,8,9-tetrasubstituted purines by a combination of the Suzuki cross-coupling, N-arylation, and direct C-H arylation reactions. Journal of Organic Chemistry 2008, 73(22), 9048 - 9054, 10.1021/jo8018126 .
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Hocek, Michal;
Klecka, Martin;
Pohl, Radek;
Klepetaova, Blanka, Direct C-H borylation and C-H arylation of pyrrolo2,3-dpyrimidines: Synthesis of 6,8-disubstituted 7-deazapurines. Organic and Biomolecular Chemistry 2009, 7(5), 866 - 868, 10.1039/b900218a .
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Hocek, Michal;
Pohl, Radek;
Vrabel, Milan;
Havran, Ludek;
Fojta, Miroslav;
Cahova, Hana;
Horakova, Petra;
Pivonkovas, Hana;
Kalachova, Lubica;
Cernocka, Hana;
Sebest, Peter, Base-modified DNA labeled by [Ru(bpy)] and [Os(bpy)] complexes: Construction by polymerase incorporation of modified nucleoside triphosphates, electrochemical and luminescent properties, and applications. Chemistry - A European Journal 2009, 15(5), 1144 - 1154, 10.1002/chem.200801538 .
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Hocek, Michal;
Pohl, Radek;
Kalachova, Lubica, Synthesis of 2′-deoxyuridine and 2′-deoxycytidine Nucleosides bearing bipyridine and terpyridine ligands at position 5. Synthesis 2009(1), 105 - 112, 10.1055/s-0028-1083266 .
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Hocek, Michal;
Pohl, Radek;
Stefko, Martin, Synthesis of benzamide-C-ribonucleosides by Pd-catalyzed aminocarbonylations. Tetrahedron 2009, 65(23), 4471 - 4483, 10.1016/j.tet.2009.04.006 .
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Hocek, Michal;
Pohl, Radek;
Havran, Ludek;
Fojta, Miroslav;
Horakova, Petra;
Sebest, Peter;
Riedl, Jan, Tetrathiafulvalene-labelled nucleosides and nucleoside triphosphates: Synthesis, electrochemistry and the scope of their polymerase incorporation into DNA. European Journal of Organic Chemistry 2009(21), 3519 - 3525, 10.1002/ejoc200900392 .
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Hocek, Michal;
Pohl, Radek;
Cernova, Miroslava, Switching the regioselectivity of direct C-H arylation of 1,3-Dimethyluracil. European Journal of Organic Chemistry 2009(22), 3698 - 3701, 10.1002/ejoc.200900586 .
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Hocek, Michal;
Pohl, Radek;
Hasnik, Zbynek, Cross-coupling reactions of halopurines with aryl- and alkyltrifluoroborates; the scope and limitations in the synthesis of modified purines. Synthesis 2009(8), 1309 - 1317, 10.1055/s-0028-1088038 .
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Hocek, Michal;
Pohl, Radek;
Klepetarova, Blanka;
Hasnik, Zbynek, Synthesis of (purin-6-yl)acetates and their transformations to 6-(2-hydroxyethyl)-and 6-(carbamoylmethyl)purines. Collect. Czech. Chem. Commun. 2009, 74(7-8), 1035 - 1059, 10.1135/cccc2009042 .
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Naus, Petr;
Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Mackman, Richard;
Dzubak, Petr;
Hajduch, Marian;
Ameral, Ria;
Birkus, Gabriel;
Wang, Ting;
Ray, Adrian S.;
Cihlar, Tomas, 6-(Het)aryl-7-deazapurine ribonucleosides as novel potent cytostatic agents. Journal of Medicinal Chemistry 2010, 53(1), 460 - 470, 10.1021/jm901428k .
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Sanda, Miloslav;
Hocek, Michal;
Pohl, Radek;
Raindlova, Veronika, Direct polymerase synthesis of reactive aldehyde-functionalized DNA and Its conjugation and staining with hydrazines. Angewandte Chemie - International Edition 2010, 49(6), 1064 - 1066, 10.1002/anie.200905556 .
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Hocek, Michal;
Pohl, Radek;
Ikonen, Satu;
MacIkova-Cahova, Hana;
Anda, Miloslav, Synthesis of nucleoside and nucleotide conjugates of bile acids, and polymerase construction of bile acid-functionalized DNA. Organic and Biomolecular Chemistry 2010, 8(5), 1194 - 1201, 10.1039/b924072a .
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Hocek, Michal;
Pohl, Radek;
Hasnik, Zbynek, Synthesis of (purin-6-yl)methylphosphonate bases and nucleosides. Tetrahedron Letters 2010, 51(18), 2464 - 2466, 10.1016/j.tetlet.2010.02.167 .
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Hocek, Michal;
Pohl, Radek;
Klepetarova, Blanka;
Cerna, Igor, Intramolecular direct C-H arylation approach to fused purines. Synthesis of purino[8, 9-f]phenanthridines and 5, 6-dihydropurino[8, 9-a]isoquinolines. Journal of Organic Chemistry 2010, 75(7), 2302 - 2308, 10.1021/jo100111t .
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Naus, Petr;
Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Ameral, Ria;
Birkus, Gabriel;
Cihlar, Tomas;
Spacilova, Pavla;
Snasel, Jan;
Zabranska, Helena;
Pichova, Iva, CycloSal-phosphate pronucleotides of cytostatic 6-(het)aryl-7-deazapurine ribonucleosides: Synthesis, cytostatic activity, and inhibition of adenosine kinases. ChemMedChem 2010, 5(8), 1386 - 1396, 10.1002/cmdc.201000192 .
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Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Birkus, Gabriel;
Cihlar, Tomas;
Perlikova, Pavla;
Shih, Robert, Phosphoramidate pronucleotides of cytostatic 6-aryl-7-deazapurine ribonucleosides. Bioorganic and Medicinal Chemistry 2011, 19(1), 229 - 242, 10.1016/j.bmc.2010.11.029 .
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Hocek, Michal;
Pohl, Radek;
Havran, Ludek;
Fojta, Miroslav;
Horakova, Petra;
Macickova-Cahova, Hana;
Spacek, Jan, Alkylsulfanylphenyl derivatives of cytosine and 7-deazaadenine nucleosides, nucleotides and nucleoside triphosphates: Synthesis, polymerase incorporation to DNA and electrochemical study. Chemistry - A European Journal 2011, 17(21), 5833 - 5841, 10.1002/chem.201003496 .
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Hocek, Michal;
Pohl, Radek;
Kielkowski, Pavel, Synthesis of acetylene linked double-nucleobase nucleos(t)ide building blocks and polymerase construction of DNA containing cytosines in the major groove. Journal of Organic Chemistry 2011, 76(9), 3457 - 3462, 10.1021/jo200436j .
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Hocek, Michal;
Pohl, Radek;
Cerna, Igor;
Cernova, Miroslava, Regioselective direct C-H arylations of protected uracils. Synthesis of 5- and 6-aryluracil bases. Journal of Organic Chemistry 2011, 76(13), 5309 - 5319, 10.1021/jo2006494 .
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Naus, Petr;
Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Dzubak, Petr;
Hajduch, Marian;
Birkus, Gabriel;
Wang, Ting;
Ray, Adrian S.;
Cihlar, Tomas;
Pichova, Iva;
Perlikova, Pavla;
Bourderioux, Aurelie;
Konecny, Petr;
Stray, Kirsten M.;
Feng, Joy Y., Synthesis and significant cytostatic activity of 7-hetaryl-7- deazaadenosines. Journal of Medicinal Chemistry 2011, 54(15), 5498 - 5507, 10.1021/jm2005173 .
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Hocek, Michal;
Pohl, Radek;
Macickova-Cahova, Hana;
Kielkowski, Pavel, Transient and switchable (Triethylsilyl)ethynyl protection of DNA against cleavage by restriction endonucleases. Angewandte Chemie - International Edition 2011, 50(37), 8727 - 8730, 10.1002/anie.201102898 .
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Hocek, Michal;
Pohl, Radek;
Havran, Ludek;
Fojta, Miroslav;
Horakova, Petra;
Balintova, Jana;
Vidlakova, Pavlina, Anthraquinone as a redox label for DNA: Synthesis, enzymatic incorporation, and electrochemistry of anthraquinone-modified nucleosides, nucleotides, and DNA. Chemistry - A European Journal 2011, 17(50), 14063 - 14073, 10.1002/chem.201101883 .
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Hocek, Michal;
Pohl, Radek;
Kalachova, Lubica, Synthesis of nucleoside mono- and triphosphates bearing oligopyridine ligands, their incorporation into DNA and complexation with transition metals. Organic and Biomolecular Chemistry 2012, 10(1), 49 - 55, 10.1039/c1ob06359f .
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Hocek, Michal;
Pohl, Radek;
Rulisek, Lubomir;
Riedl, Jan, Synthesis and photophysical properties of biaryl-substituted nucleos(t)ides. Polymerase synthesis of DNA probes bearing solvatochromic and pH-sensitive dual fluorescent and F NMR labels. Journal of Organic Chemistry 2012, 77(2), 1026 - 1044, 10.1021/jo202321g .
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Hocek, Michal;
Pohl, Radek;
Joubert, Nicolas;
Kubelka, Tomas;
Chapuis, Hubert, Synthesis of 6-substituted 2(1H)-pyridon-3-yl C-2′- deoxyribonucleosides. European Journal of Organic Chemistry 2012(9), 1759 - 1767, 10.1002/ejoc.201101662 .
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Hocek, Michal;
Pohl, Radek;
Raindlova, Veronika, Synthesis of aldehyde-linked nucleotides and DNA and their bioconjugations with lysine and peptides through reductive amination. Chemistry - A European Journal 2012, 18(13), 4080 - 4087, 10.1002/chem.201103270 .
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Naus, Petr;
Hocek, Michal;
Pohl, Radek;
Perlikova, Pavla, Sugar-modified derivatives of cytostatic 6-(het)aryl-7-deazapurine nucleosides: 2′-c-methylribonucleosides, arabinonucleosides and 2′-deoxy-2′-fluoroarabinonucleosides. Collect. Czech. Chem. Commun. 2011, 76(8), 957 - 988, 10.1135/cccc2011082 .
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Hocek, Michal;
Pohl, Radek;
Klepetarova, Blanka;
Cernova, Miroslava, A general regioselective synthesis of 2,4-diarylpyrimidines from 2-thiouracil through two orthogonal cross-coupling reactions. Synlett 2012, 23(9), 1305 - 1308, 10.1055/s-0031-1290826 .
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Naus, Petr;
Hocek, Michal;
Votruba, Ivan;
Pohl, Radek;
Slavetinska, Lenka;
Birkus, Gabriel;
Cihlar, Tomas;
Perlikova, Pavla;
Bourderioux, Aurelie;
Bahador, Gina, Sugar-modified derivatives of cytostatic 7-(het)aryl-7-deazaadenosines: 2′-C-methylribonucleosides, 2′-deoxy-2′- fluoroarabinonucleosides, arabinonucleosides and 2′-deoxyribonucleosides. Bioorganic and Medicinal Chemistry 2012, 20(17), 5202 - 5214, 10.1016/j.bmc.2012.07.003 .
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Hocek, Michal;
Pohl, Radek;
Tichy, Michal;
Xu, Hao Ying;
Chen, Yen-Liang;
Yokokawa, Fumiaki;
Shi, Pei-Yong, Synthesis and antiviral activity of 4,6-disubstituted pyrimido[4,5-b]indole ribonucleosides. Bioorganic and Medicinal Chemistry 2012, 20(20), 6123 - 6133,11, 10.1016/j.bmc.2012.08.021 .
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Hocek, Michal;
Pohl, Radek;
Macickova-Cahova, Hana, Cleavage of Functionalized DNA Containing 5-Modified Pyrimidines by Type II Restriction Endonucleases. Chembiochem : a European journal of chemical biology 2011, 12(3), 431 - 438, 10.1002/cbic.201000644 .
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Hocek, Michal;
Pohl, Radek;
Fojta, Miroslav;
Ernsting, Nikolaus P.;
Riedl, Jan;
Orsag, Petr, Labelling of nucleosides and oligonucleotides by solvatochromic 4-aminophthalimide fluorophore for studying DNA-protein interactions. Chemical Science 2012, 3(9), 2797 - 2806, 10.1039/c2sc20404e .
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Hocek, Michal;
Pohl, Radek;
Klepetarova, Blanka;
Havran, Ludek;
Fojta, Miroslav;
Pivonkova, Hana;
Horakova, Petra;
Raindlova, Veronika;
Simkov, Eva, Synthesis of hydrazone-modified nucleotides and their polymerase incorporation onto DNA for redox labeling. ChemPlusChem 2012, 77(8), 652 - 662, 10.1002/cplu.201200056 .
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Menova, Petra;
Hocek, Michal;
Pohl, Radek;
Fojta, Miroslav;
Riedl, Jan;
Orsag, Petr, GFP-like fluorophores as DNA labels for studying DNA-protein interactions. Journal of Organic Chemistry 2012, 77(18), 8287 - 8293, 10.1021/jo301684b .
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Hocek, Michal;
Pohl, Radek;
Bednarova, Lucie;
Kalachova, Lubica;
Fanfrlik, Jindrich, Synthesis of nucleosides and dNTPs bearing oligopyridine ligands linked through an octadiyne tether, their incorporation into DNA and complexation with transition metal cations. Organic and Biomolecular Chemistry 2013, 11(1), 78 - 89, 10.1039/c2ob26881g .
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Cejka, Jan;
Hocek, Michal;
Klecka, Martin;
Pohl, Radek, Direct C-H sulfenylation of purines and deazapurines. Organic and Biomolecular Chemistry 2013, 11(31), 5189 - 5193, 10.1039/c3ob40881g .
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Hocek, Michal;
Pohl, Radek;
Bahador, Gina;
Tichy, Michal;
Lee, Yu-Jen;
Tloust'Ova, Eva;
Weber, Jan, Synthesis and biological activity of benzo-fused 7-deazaadenosine analogues. 5- and 6-substituted 4-amino- or 4-alkylpyrimido[4,5-b]indole ribonucleosides. Bioorganic and Medicinal Chemistry 2013, 21(17), 5362 - 5372, 10.1016/j.bmc.2013.06.011 .
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Hocek, Michal;
Pohl, Radek;
Havran, Ludek;
Fojta, Miroslav;
Balintova, Jana;
Vidlakova, Pavlina;
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